[Other] Utilizing Molecular Dynamics and Mechanistic Pharmacokinetic Studies in the Design of Selective CDK2 Inhibitors

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journal:Journal of Medicinal Chemistry

Authors:Vishal A. Verma; Jessica M. Grandner; Brendan T. Parr; Mingshuo Zeng; Melissa Ashley; Yong Wang; Paul Beroza; Pasquale Carione; Kevin M. Johnson; Angela J. Oh; Jeremy M. Murray; James R. Kiefer; John G. Moffat; Madeleine Prangley; Karl Merrick; Steffan Vartanian; Marc Hafner; Christine J. Orr; Ehud Segal; Elizabeth S. Levy; Jian Wang; Zijin Xu; Shouliang Wang; Guijun Liu; Yanan Niu; Xufeng Li; Qisen Zhang; Zebin Ma; Mingyan Sun; Zengyang Wu; Wanqiu Zhao; Ye Li; Lina Zhang; Steven R. Magnuson; Karen E. Samy

Published date:--

DOI:10.1021/acs.jmedchem.5c03803

PDF link:https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c03803

Article link:https://doi.org/10.1021/acs.jmedchem.5c03803

Article Source:American Chemical Society (ACS)


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