[ACS] Development of Orally Bioavailable Peptides Targeting an Intracellular Protein: From a Hit to a Clinical KRAS Inhibitor

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journalㄩJournal of the American Chemical Society

AuthorsㄩMikimasa Tanada; Minoru Tamiya; Atsushi Matsuo; Aya Chiyoda; Koji Takano; Toshiya Ito; Machiko Irie; Tomoya Kotake; Ryuuichi Takeyama; Hatsuo Kawada; Ryuji Hayashi; Shiho Ishikawa; Kenichi Nomura; Noriyuki Furuichi; Yuya Morita; Mirai Kage; Satoshi Hashimoto; Keiji Nii; Hitoshi Sase; Kazuhiro Ohara; Atsushi Ohta; Shino Kuramoto; Yoshikazu Nishimura; Hitoshi Iikura; Takuya Shiraishi

Published dateㄩ2023-8-2

DOIㄩ10.1021/jacs.3c03886

PDF linkㄩhttps://pubs.acs.org/doi/pdf/10.1021/jacs.3c03886

Article linkㄩhttps://doi.org/10.1021/jacs.3c03886

Article SourceㄩAmerican Chemical Society (ACS)


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